pK i values | |||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|
Receptors Ligands | α2- | D2-like | 5-HT1 | ||||||||
α 2A | α 2B | α 2C | D2 | D3 | D4 | 1Aª | 1B | 1D | 1E | 1F | |
DHE | 8.7a | 8.0a | 9.0a | 8.2a | 8.2a | 8.1a | 9.3a | (r)7.8a | 8.6a | 6.2a | 6.9a |
Rauwolscine | 8.9b | 8.9b | 9.3b | N.D. | N.D. | 6.5c | 7.8c | 5.5c | N.D. | ||
GR127935 | < 6.0 d,* | N.D. | 7.2 e | (r)8.8f | 8.6g | 5.4g | 6.4g | ||||
Haloperidol | 5.8 h,* | 9.4i | 8.5i | 8.8i | N.D. |